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Diversity oriented clicking delivers β-substituted alkenyl sulfonyl fluorides as covalent human neutrophil elastase inhibitors
https://www.pnas.org/doi/10.1073/pnas.2208540119#fig01

First corresponding paper on bioRxiv! PROTAC-mediated selective degradation of cytosolic soluble epoxide hydrolase enhances ER-stress reduction #3
https://www.biorxiv.org/content/10.1101/2022.01.20.477134v1
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